GSK-923295

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TargetMol
Product Code: TAR-T2039
Supplier: TargetMol
CodeSizePrice
TAR-T2039-1mg1mg£107.00
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TAR-T2039-2mg2mg£122.00
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TAR-T2039-5mg5mg£149.00
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TAR-T2039-1mL1 mL * 10 mM (in DMSO)£181.00
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TAR-T2039-10mg10mg£213.00
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TAR-T2039-25mg25mg£351.00
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TAR-T2039-50mg50mg£502.00
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TAR-T2039-100mg100mg£693.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).
CAS:
1088965-37-0
Formula:
C32H38ClN5O4
Molecular Weight:
592.14
Pathway:
Cytoskeletal Signaling; Apoptosis
Purity:
0.9971
SMILES:
CC(C)Oc1ccc(cc1Cl)C(=O)N[C@H](CNC(=O)CN(C)C)Cc1ccc(cc1)-c1cn2cccc([C@H](C)O)c2n1
Target:
Apoptosis; Kinesin

References

1. Wood KW, et al. Proc Natl Acad Sci U S A, 2010, 107(13), 5839-5844. 2. Qian XP, et al. ACS Med Chem Lett, 2010, 1, 30?34. 3. Lock RB, et al. Pediatr Blood Cancer 2012, 58(6), 916?923. 4. Mayes PA, et al. Int J Cancer, 2013, 132(3), E149-157.