Deltarasin

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TargetMol
Product Code: TAR-T6462
Supplier: TargetMol
CodeSizePrice
TAR-T6462-25mg25mgEnquire
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TAR-T6462-50mg50mgEnquire
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TAR-T6462-1mg1mg£103.00
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TAR-T6462-2mg2mg£118.00
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TAR-T6462-5mg5mg£168.00
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TAR-T6462-1mL1 mL * 10 mM (in DMSO)£201.00
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TAR-T6462-10mg10mg£229.00
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Deltarasin is a small molecular inhibitor of KRAS-PDEδ interaction with Kd of 38 nM for binding to purified PDEδ.
CAS:
1440898-61-2
Formula:
C40H37N5O
Molecular Weight:
603.77
Pathway:
Metabolism; GPCR/G Protein; MAPK
Purity:
0.9906
SMILES:
C(Oc1ccc(cc1)-c1nc2ccccc2n1Cc1ccccc1)[C@H](C1CCNCC1)n1c(nc2ccccc12)-c1ccccc1
Target:
PDE; Ras

References

Zimmermann G, et al. Nature. 2013, 497(7451), 638-642.