Encenicline
Code | Size | Price |
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TAR-T7193-1mg | 1mg | £160.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-2mg | 2mg | £205.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-5mg | 5mg | £262.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-1mL | 1 mL * 10 mM (in DMSO) | £278.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-10mg | 10mg | £380.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-25mg | 25mg | £589.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-50mg | 50mg | £809.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7193-100mg | 100mg | £1,075.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Encenicline is a selective α7 nicotinic acetylcholine receptor (nAChRs) agonist in development for treating cognitive impairment in schizophrenia and Alzheimer's disease.
CAS:
550999-75-2
Formula:
C16H17ClN2OS
Molecular Weight:
320.84
Pathway:
Neuroscience
Purity:
0.98
SMILES:
Clc1cccc2cc(sc12)C(=O)N[C@H]1CN2CCC1CC2
Target:
AChR
References
Prickaerts J, van Goethem NP, Chesworth R,et al.EVP-6124, a novel and selective ?7 nicotinic acetylcholine receptor partial agonist, improves memory performance by potentiating the acetylcholine response of ?7 nicotinic acetylcholine receptors[J].Neuropharmacology. 2012 Feb;62(2):1099-110.
Hayward A , Adamson L , Neill J C . Partial agonism at the ?7 nicotinic acetylcholine receptor improves attention, impulsive action and vigilance in low attentive rats[J]. European Neuropsychopharmacology, 2017, 27(4):325-335.