(E)-SI-2

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TargetMol
Product Code: TAR-T9836
Supplier: TargetMol
CodeSizePrice
TAR-T9836-1mg1mg£189.00
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TAR-T9836-5mg5mg£340.00
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Quantity:
TAR-T9836-1mL1 mL * 10 mM (in DMSO)£346.00
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Quantity:
TAR-T9836-10mg10mg£470.00
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Quantity:
TAR-T9836-25mg25mg£707.00
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Quantity:
TAR-T9836-50mg50mg£978.00
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Quantity:
TAR-T9836-100mg100mg£1,291.00
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Quantity:
TAR-T9836-500mg500mg£2,456.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Documents

Further Information

Bioactivity:
(E)-SI-2 is a potent small-molecule inhibitor of steroid receptor coactivator-3 (SRC-3 or AIB1) that can selectively inhibit the intrinsic transcriptional activities of SRC-3, also inhibits SRC-1 and SRC-2. It selectively reduces cellular protein levels of SRC-3, but not that of CARM-1, blocks MDA-MB-468 cell growth with an IC50 value of 3.4 nM, but spares normal cells.
CAS:
380537-35-9
Formula:
C15H15N5
Molecular Weight:
265.31
Purity:
0.98
SMILES:
CN1C2=CC=CC=C2N=C1N/N=C(C3=NC=CC=C3)C