Aaptamine
Code | Size | Price |
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TAR-TN1354-1mL | 1 mL * 10 mM (in DMSO) | £384.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-TN1354-10mg | 10mg | £512.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Aaptamine functions as a proteasome inhibitor, it activates p21 promoter in a p53-independent manner.
CAS:
85547-22-4
Formula:
C13H12N2O2
Molecular Weight:
228.251
Pathway:
Cell Cycle/Checkpoint; Apoptosis
Purity:
0.98
SMILES:
COc1cc2ccnc3cc[nH]c(c1OC)c23
Target:
c-Myc; TNF; p53
References
Activity of aaptamine and two derivatives, demethyloxyaaptamine and isoaaptamine, in cisplatin-resistant germ cell cancer.J Proteomics. 2014 Jan 16;96:223-39.