[Orn5]-URP

TargetMol
Product Code: TAR-TP1928
Supplier: TargetMol
CodeSizePrice
TAR-TP1928-1mg1mg£186.00
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Urotensin-II (UT) receptor pure antagonist (pEC50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay.
CAS:
782485-03-4
Formula:
C48H62N10O10S2
Molecular Weight:
1003.2
Purity:
0.98
SMILES:
0

References

Chatenet et al (2004) Structure-activity relationships and structural conformation of a novel urotensin II-related peptide. Peptides 25 1819 PMID: Diallo et al (2008) [Orn5]URP acts as a pure antagonist of urotensinergic receptors in rat cortical astrocytes. Peptides 29 813 PMID: