PG106

TargetMol
Product Code: TAR-TP1952
Supplier: TargetMol
CodeSizePrice
TAR-TP1952-1mg1mg£294.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

1 / 1

Further Information

Bioactivity:
Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.
CAS:
944111-22-2
Formula:
C51H69N13O9
Molecular Weight:
1008.19
Purity:
0.98
SMILES:
0

References

Grieco et al (2007) Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: their activity and selectivity at human melanocortin receptors 3, 4, and 5. Peptides. 28 1191 PMID: