XMD8-87

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TargetMol
Product Code: TAR-T3709
Supplier: TargetMol
CodeSizePrice
TAR-T3709-2mg2mg£102.00
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TAR-T3709-5mg5mg£128.00
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TAR-T3709-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T3709-10mg10mg£172.00
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TAR-T3709-25mg25mg£298.00
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TAR-T3709-50mg50mg£436.00
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TAR-T3709-100mg100mg£610.00
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TAR-T3709-500mg500mg£1,219.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
XMD8-87 is a TNK2 inhibitor with activity in the inhibition of TNK2 phosphorylation. XMD8-87 and XMD16-5 potently inhibit phosphorylation of TNK2 truncation mutations found in solid tumor types.
CAS:
1234480-46-6
Formula:
C24H27N7O2
Molecular Weight:
445.527
Pathway:
DNA Damage/DNA Repair; Metabolism; Proteases/Proteasome
Purity:
0.9761
SMILES:
COc1cc(ccc1Nc1ncc2NC(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1
Target:
Tyrosinase; PPAR

References

Maxson JE, et al. Cancer Res. 2016, 76(1):127-38.