CCT128930

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TargetMol
Product Code: TAR-T6303
Supplier: TargetMol
CodeSizePrice
TAR-T6303-1mg1mg£108.00
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TAR-T6303-2mg2mg£123.00
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TAR-T6303-1mL1 mL * 10 mM (in DMSO)£164.00
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TAR-T6303-5mg5mg£164.00
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TAR-T6303-10mg10mg£238.00
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TAR-T6303-25mg25mg£399.00
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TAR-T6303-50mg50mg£548.00
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TAR-T6303-100mg100mg£766.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CCT128930 is a potent, ATP-competitive and selective inhibitor of Akt2 with IC50 of 6 nM, 28-fold greater selectivity for Akt2 than the closely related PKA kinase.
CAS:
885499-61-6
Formula:
C18H20ClN5
Molecular Weight:
341.84
Pathway:
MAPK; Autophagy; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Purity:
0.9918
SMILES:
NC1(Cc2ccc(Cl)cc2)CCN(CC1)c1ncnc2[nH]ccc12
Target:
Akt; PKA; S6 Kinase; Autophagy

References

Yap TA, et al. Mol Cancer Ther. 2011, 10(2), 360-371.