KRN5

TargetMol
Product Code: TAR-T13747
Supplier: TargetMol
CodeSizePrice
TAR-T13747-5mg5mg£850.00
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Quantity:
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
KRN5 is an effective inhibitor of NFAT5 with an IC50 of 750 nM and can be used in studies about chronic arthritis.
CAS:
1800465-47-7
Formula:
C27H22FNO5
Molecular Weight:
459.47
Purity:
0.9882
SMILES:
O=C1C=2C(OC)=C(OC)C=CC2C(=C3C4=CC=5OCOC5C=C4CCN13)CC=6C=CC=CC6F

References

1. Han EJ, et al. Suppression of NFAT5-mediated Inflammation and Chronic Arthritis by Novel ?B-binding Inhibitors. EBioMedicine. 2017 Apr;18:261-273.