Lavendustin C6
Code | Size | Price |
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TAR-T25644-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T25644-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T25644-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Lavendustin C6 is a effective tyrosine kinase inhibitor.
CAS:
144676-04-0
Formula:
C20H25NO5
Molecular Weight:
359.422
Purity:
0.98
SMILES:
CCCCCCN(Cc1cc(O)ccc1O)c1ccc(O)c(c1)C(O)=O
References
1. Yoon J, Ryu JS. A rapid synthesis of lavendustin-mimetic small molecules by click fragment assembly. Bioorg Med Chem Lett. 2010 Jul 1;20(13):3930-5. doi: 10.1016/j.bmcl.2010.05.014. Epub 2010 May 12. PubMed PMID: 20570145.
2. Agbotounou WK, Umezawa K, Jacquemin-Sablon A, Pierre J. Inhibition by two lavendustins of the tyrosine kinase activity of pp60F527 in vitro and in intact cells. Eur J Pharmacol. 1994 Sep 15;269(1):1-8. PubMed PMID: 7828651.
3. Nynca A, Nynca J, W?sowska B, Kolesarova A, Ko?omycka A, Ciereszko RE. Effects of the phytoestrogen, genistein, and protein tyrosine kinase inhibitor-dependent mechanisms on steroidogenesis and estrogen receptor expression in porcine granulosa cells of medium follicles. Domest Anim Endocrinol. 2013 Jan;44(1):10-8. doi: 10.1016/j.domaniend.2012.07.002. Epub 2012 Aug 10. PubMed PMID: 22920265.
4. Kobayashi T, Nemoto S, Ishida K, Taguchi K, Matsumoto T, Kamata K. Involvement of CaM kinase II in the impairment of endothelial function and eNOS activity in aortas of Type 2 diabetic rats. Clin Sci (Lond). 2012 Sep;123(6):375-86. doi: 10.1042/CS20110621. PubMed PMID: 22494112.