RGH 1756
Code | Size | Price |
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TAR-T26069-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26069-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26069-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.
CAS:
207277-37-0
Formula:
C26H30N4O2S
Molecular Weight:
462.61
Purity:
0.98
SMILES:
COc1ccccc1N1CCN(CCCCOc2ccc(cc2)-c2cn3ccsc3n2)CC1
References
1. G?mesi LI, Kap?s M, Szeber?nyi S. Application of LC-MS analysis to the characterisation of the in vitro and in vivo metabolite profiles of RGH-1756 in the rat. J Pharm Biomed Anal. 2001 Mar;24(5-6):877-85. PubMed PMID: 11248481.
2. Kov?cs KJ, Csejtei M, Laszlovszky I. Double activity imaging reveals distinct cellular targets of haloperidol, clozapine and dopamine D(3) receptor selective RGH-1756. Neuropharmacology. 2001 Mar;40(3):383-93. PubMed PMID: 11166331.
3. S?v?g? J, Farde L, Halldin C, Schukin E, Schou M, Laszlovszky I, Kiss B, Guly?s B. Lack of effect of reserpine-induced dopamine depletion on the binding of the dopamine-D3 selective radioligand, [11C]RGH-1756. Brain Res Bull. 2005 Oct 15;67(3):219-24. PubMed PMID: 16144658.
4. Terj?ki E, Kap?s M. An HPLC/UV method for the determination of RGH-1756 in dog and rat plasma. J Pharm Biomed Anal. 2001 Mar;24(5-6):913-20. PubMed PMID: 11248484.