Risotilide
Code | Size | Price |
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TAR-T26092-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26092-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T26092-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.
CAS:
120688-08-6
Formula:
C15H27N3O4S2
Molecular Weight:
377.52
Purity:
0.98
SMILES:
CC(C)NCCN(C(C)C)S(=O)(=O)c1ccc(NS(C)(=O)=O)cc1
References
1. Hewett KW, Le FK, Martin KL, Brasington CR, Piecuch S, Case CL. Changes in atrioventricular conduction properties with refractory-period modulation. J Cardiovasc Pharmacol. 1996 Dec;28(6):824-32. PubMed PMID: 8961081.
2. McLarnon JG, Wang XP. Actions of cardiac drugs on a calcium-dependent potassium channel in hippocampal neurons. Mol Pharmacol. 1991 Apr;39(4):540-6. PubMed PMID: 2017153.
3. Kowey PR, Friechling TD, Sewter J, Wu Y, Sokil A, Paul J, Nocella J. Electrophysiological effects of left ventricular hypertrophy. Effect of calcium and potassium channel blockade. Circulation. 1991 Jun;83(6):2067-75. PubMed PMID: 1645624.
4. Burckhardt BC, G?gelein H. Small and maxi K+ channels in the basolateral membrane of isolated crypts from rat distal colon: single-channel and slow whole-cell recordings. Pflugers Arch. 1992 Jan;420(1):54-60. PubMed PMID: 1553263.