CV-1674
| Code | Size | Price |
|---|
| TAR-T31115-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
| TAR-T31115-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
| TAR-T31115-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
CV-1674 induced selective coronary vasodilation and had little effect on cardiac hemodynamics.
CAS:
37151-17-0
Formula:
C17H19N5O5
Molecular Weight:
373.369
Purity:
0.98
SMILES:
COc1ccc(cc1)-c1nc(N)c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
References
1. Hirata M, Kawazoe K, Tanabe M, Kikuchi K. Effects of a 2-substituted adenosine derivative, 2-(p-methoxyphenyl)-adenosine (CV-1674) on coronary and cardiohemodynamics, and myocardial energetics. Jpn J Pharmacol. 1977 Oct;27(5):689-700. PubMed PMID: 592558.
2. Singh YN, Dryden WF, Chen H. The inhibitory effects of some adenosine analogues on transmitter release at the mammalian neuromuscular junction. Can J Physiol Pharmacol. 1986 Nov;64(11):1446-50. PubMed PMID: 3024786.
3. Paton DM. Presynaptic inhibition of neurotransmission in rat vas deferens by 2-(p-methoxyphenyl) adenosine, ethyl adenosine-5'-carboxylate and N-cyclopropyl adenosine-5'-carboxamide. J Pharm Pharmacol. 1980 Feb;32(2):133-5. PubMed PMID: 6103035.
4. van der Ploeg I, Ahlberg S, Parkinson FE, Olsson RA, Fredholm BB. Functional characterization of adenosine A2 receptors in Jurkat cells and PC12 cells using adenosine receptor agonists. Naunyn Schmiedebergs Arch Pharmacol. 1996 Feb;353(3):250-60. PubMed PMID: 8692279.