GYKI-53405
Code | Size | Price |
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TAR-T32034-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T32034-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T32034-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
GYKI-53405 (LY 293606) is a non-competitive AMPA receptor antagonist.
CAS:
143691-37-6
Formula:
C19H19N3O3
Molecular Weight:
337.379
Purity:
0.98
SMILES:
CC1Cc2cc3OCOc3cc2C(=NN1C(C)=O)c1ccc(N)cc1
References
1. Jakus R, Graf M, Ando RD, Balogh B, Gacsalyi I, Levay G, Kantor S, Bagdy G. Effect of two noncompetitive AMPA receptor antagonists GYKI 52466 and GYKI 53405 on vigilance, behavior and spike-wave discharges in a genetic rat model of absence epilepsy. Brain Res. 2004 May 22;1008(2):236-44. PubMed PMID: 15145761.
2. Szabados T, Gigler G, Gacs?lyi I, Gyerty?n I, L?vay G. Comparison of anticonvulsive and acute neuroprotective activity of three 2,3-benzodiazepine compounds, GYKI 52466, GYKI 53405, and GYKI 53655. Brain Res Bull. 2001 Jun;55(3):387-91. PubMed PMID: 11489346.
3. Szab? G, Henley JM. Binding of the AMPA receptor antagonist [3H]GYKI 53405 to Xenopus brain membranes. Neuroreport. 1993 Oct 25;5(1):93-4. PubMed PMID: 7506593.