BMS-986121
Code | Size | Price |
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TAR-T40392-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T40392-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
BMS-986121 is a positive allosteric modulator (PAM) of the μ opioid receptor extracted from patent WO2014107344. BMS-986121 is built on a chemical scaffold representing a new chemotype for μ receptor PAMs.
CAS:
313671-26-0
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
WO2014107344
Bisignano P, et al. Ligand-Based Discovery of a New Scaffold for Allosteric Modulation of the ?-Opioid Receptor. J Chem Inf Model. 2015;55(9):1836-1843.
Burford NT, et al. Discovery of positive allosteric modulators and silent allosteric modulators of the ?-opioid receptor. Proc Natl Acad Sci U S A. 2013;110(26):10830-10835.