Prucalopride

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TargetMol
Product Code: TAR-T2542
Supplier: TargetMol
CodeSizePrice
TAR-T2542-5mg5mg£96.00
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Quantity:
TAR-T2542-1mL1 mL * 10 mM (in DMSO)£110.00
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Quantity:
TAR-T2542-10mg10mg£112.00
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Quantity:
TAR-T2542-25mg25mg£125.00
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Quantity:
TAR-T2542-50mg50mg£136.00
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TAR-T2542-100mg100mg£183.00
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TAR-T2542-200mg200mg£230.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Prucalopride is a selective, high-affinity 5-HT4A/4B receptor agonist (Ki: 2.5/8 nM). It has >290-fold selectivity for 5-HT4A/4B receptor than other 5-HT receptor subtypes.
CAS:
179474-81-8
Formula:
C18H26ClN3O3
Molecular Weight:
367.87
Pathway:
GPCR/G Protein; Neuroscience
Purity:
1
SMILES:
COCCCN1CCC(CC1)NC(=O)c1cc(Cl)c(N)c2CCOc12
Target:
5-HT Receptor

References

1. Briejer MR, et al. Eur J Pharmacol, 2001, 423(1), 71-83. 2. Camilleri M, et al. N Engl J Med, 2008, 358(22), 2344-2354. 3. Bouras EP, et al. Gastroenterology, 2001, 120(2), 354-360. 4. Tack J, et al. Gut, 2009, 58(3), 357-365. 5. Briejer MR, et al. Neurogastroenterol Motil, 2001, 13(5), 465-472.