BCAT-IN-1
Code | Size | Price |
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TAR-T40218-25mg | 25mg | £1,099.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T40218-50mg | 50mg | £1,669.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T40218-100mg | 100mg | £2,464.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
BCAT-IN-1 is a potent, selective and orally active inhibitor of BCATm , with a pIC 50 of 7.3. BCAT-IN-1 shows 100-fold selectivity for BCATm over BCATc ( pIC 50 =5.4). BCAT-IN-1 can be used for the research of metabolic diseases.
CAS:
2581243-32-3
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0
References
Deng H, et, al. Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2-Aryl Benzimidazole BCATm Inhibitors. ACS Med Chem Lett. 2016 Feb 8;7(4):379-84.