YIL 781
Code | Size | Price |
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TAR-T23543-1mg | 1mg | £106.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T23543-5mg | 5mg | £148.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T23543-1mL | 1 mL * 10 mM (in DMSO) | £171.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T23543-10mg | 10mg | £195.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T23543-25mg | 25mg | £334.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T23543-50mg | 50mg | £466.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T23543-100mg | 100mg | £624.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Ghrelin receptor antagonist
CAS:
875258-85-8
Formula:
C24H28FN3O2?HCl
Molecular Weight:
445.96
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
FC1=CC=C(C=C1)OC2=CC=C3N=C(C)N(C(C3=C2)=O)C[C@@H]4CN(C(C)C)CCC4.Cl
Target:
GHSR
References
Kawamura K, et al. Developing new PET tracers to image the growth hormone secretagogue receptor 1a (GHS-R1a). Nucl Med Biol. 2017;52:49-56.
Liu S, Li B, Qin B. Ghrelin protects retinal ganglion cells against rotenone via inhibiting apoptosis, restoring mitochondrial function, and activating AKT-mTOR signaling. Neuropeptides. 2018;67:63-70.
Mende F, et al. Translating biased signaling in the ghrelin receptor system into differential in vivo functions. Proc Natl Acad Sci U S A. 2018;115(43):10255-10264.
Sim YB, al. Ghrelin administered spinally increases the blood glucose level in mice. Peptides. 2014;54:162-165.