(R)-STU104
Code | Size | Price |
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TAR-T60657-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T60657-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T60657-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
(R)-STU104 is a potent and orally active TAK1-MKK3 interaction inhibitor that can be used in ulcerative colitis research. (R)-STU104 has IC50s of 0.58 uM and 4.0 uM for the phosphorylation of TNF-α and MKK3. (R)-STU104 binds with MKK3 and disrupts the TAK1 phosphorylating MKK3 to suppress the TAK1/MKK3/p38/MnK1/MK2/elF4E signal pathways [1].
CAS:
2767124-77-4
Molecular Weight:
298.338
Purity:
0.98
SMILES:
COc1ccc(cc1)[C@H]1CC(=O)c2cc(OC)cc(OC)c12