HDAC6 degrader-3
Code | Size | Price |
---|
TAR-T75018-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T75018-5mg | 5mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Documents
Further Information
Bioactivity:
HDAC6 degrader-3 is a potent and selective HDAC6 degrader via ternary complex formation and the ubiquitin-proteasome pathway with a DC 50 value of 19.4 nM. HDAC6 degrader-3 has IC 50 s of 4.54 nM and 0.647 uM for HDAC6 and HDAC1 , respectively. HDAC6 degrader-3 causes strong hyperacetylation of α-tubulin [1] .
CAS:
2785404-83-1
Molecular Weight:
883.8
Purity:
0.98