Y06037
Code | Size | Price |
---|
TAR-T24404-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T24404-500mg | 500mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
Y06037 is a BET inhibitor for the potential treatment of Castration-Resistant Prostate Cancer (CRPC). It potently inhibited cell growth, colony formation, and the expression of AR, AR-regulated genes and MYC in prostate cancer cell lines. Y06037 bounds to the BRD4(1) bromodomain (Kd: 81 nM).
CAS:
T24404
Formula:
C27H32N4O2
Molecular Weight:
444.58
Purity:
0.98
SMILES:
CC1=NOC2=CC=C(C3=NC4=CC=C(N5[C@@H](C)COCC5)C=C4N3CC6CCCCC6)C=C12