TargetMol

GOT1 inhibitor-1

Product Code:
 
TAR-T8766
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8766-1mg1mg£138.00
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TAR-T8766-5mg5mg£229.00
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TAR-T8766-1mL1 mL * 10 mM (in DMSO)£252.00
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TAR-T8766-10mg10mg£334.00
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TAR-T8766-25mg25mg£519.00
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TAR-T8766-50mg50mg£703.00
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Quantity:
TAR-T8766-100mg100mg£970.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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  • Further Information
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Further Information

Bioactivity:
GOT1 inhibitor-1 is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.
CAS:
732973-87-4
Formula:
C19H19ClN4O
Molecular Weight:
354.84
Purity:
0.9844
SMILES:
Clc1ccc(NC(=O)N2CCN(CC2)c2cccc3[nH]ccc23)cc1

Documents

References

Anglin J , Zavareh R B , Sander P N , et al. Discovery and optimization of aspartate aminotransferase 1 inhibitors to target redox balance in pancreatic ductal adenocarcinoma[J]. Bioorganic & Medicinal Chemistry Letters, 2018:S0960894X18303743.