TargetMol

BRL 54443

Product Code:
 
TAR-T2459
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2459-5mg5mg£109.00
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Quantity:
TAR-T2459-1mL1 mL * 10 mM (in DMSO)£114.00
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Quantity:
TAR-T2459-10mg10mg£132.00
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Quantity:
TAR-T2459-25mg25mg£199.00
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Quantity:
TAR-T2459-50mg50mg£273.00
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Quantity:
TAR-T2459-100mg100mg£410.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).
CAS:
57477-39-1
Formula:
C14H18N2O
Molecular Weight:
230.311
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9995
SMILES:
CN1CCC(CC1)c1c[nH]c2ccc(O)cc12
Target:
5-HT Receptor

References

1. Janssen P, et al. Eur J Pharmacol. 2004, 492(2-3), 259-267. 2. McKune CM, et al. J Pharmacol Exp Ther. 2001, 297(1), 88-95. 3. Xu P, Huang S, Zhang H, et al. Structural insights into the lipid and ligand regulation of serotonin receptors[J]. Nature. 2021, 592(7854): 469-473.