TargetMol

ES 6864

Product Code:
 
TAR-T25386
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25386-5mg5mg£930.00
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Quantity:
TAR-T25386-50mg50mg£1,821.00
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Quantity:
TAR-T25386-100mg100mg£2,319.00
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Further Information

Bioactivity:
ES 6864 is an orally active inhibitor of renin.
CAS:
116326-39-7
Formula:
C42H58N6O7S
Molecular Weight:
791.02
Purity:
0.98
SMILES:
OC(CC(=O)NCCN1CCOCC1)C(CC1CCCCC1)NC(=O)C(Cc1cscn1)NC(=O)C(CC(=O)N1CCOCC1)Cc1cccc2ccccc12

References

1. Hiwada K, Kokubu T, Murakami E, Muneta S, Morisawa Y, Yabe Y, Koike H, Iijima Y. A highly potent and long-acting oral inhibitor of human renin. Hypertension. 1988 Jun;11(6 Pt 2):708-12. PubMed PMID: 3134306. 2. Muneta S. [In vitro and in vivo inhibition of renin by a thiazolylalanyl cyclostatine derivative]. Nihon Jinzo Gakkai Shi. 1989 Aug;31(8):865. Japanese. PubMed PMID: 2512401. 3. Hiwada K. [Clinical application of renin inhibitors in the treatment of hypertension]. Nihon Rinsho. 1989 Sep;47(9):2041-6. Japanese. PubMed PMID: 2687512.