TargetMol

KNT-127

Product Code:
 
TAR-T25583
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25583-5mg5mg£1,026.00
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TAR-T25583-50mg50mg£2,464.00
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Quantity:
TAR-T25583-100mg100mg£3,283.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
KNT-127 is an agonist of δ-Opioid receptor.
CAS:
1256921-89-7
Formula:
C24H24N2O2
Molecular Weight:
372.468
Purity:
0.98
SMILES:
[H][C@]12Cc3ccc(O)cc3[C@@]3(CCN1C)Cc1nc4ccccc4cc1C[C@@]23O

References

1. Saitoh A, Tominaga H, Ogawa Y, Irukayama-Tomobe Y, Yamada M, Yanagisawa M, Nagase H. Effects of the delta opioid receptor agonist KNT-127 on electroencephalographic activity in mice. Pharmacol Rep. 2018 Apr;70(2):350-354. doi: 10.1016/j.pharep.2017.08.018. Epub 2017 Oct 28. PubMed PMID: 29477045. 2. Saitoh A, Suzuki S, Soda A, Ohashi M, Yamada M, Oka JI, Nagase H, Yamada M. The delta opioid receptor agonist KNT-127 in the prelimbic medial prefrontal cortex attenuates veratrine-induced anxiety-like behaviors in mice. Behav Brain Res. 2018 Jan 15;336:77-84. doi: 10.1016/j.bbr.2017.08.041. Epub 2017 Aug 31. PubMed PMID: 28864205. 3. Gotoh L, Saitoh A, Yamada M, Fujii H, Nagase H, Yamada M. Effects of repeated treatment with a delta opioid receptor agonist KNT-127 on hyperemotionality in olfactory-bulbectomized rats. Behav Brain Res. 2017 Apr 14;323:11-14. doi: 10.1016/j.bbr.2016.11.008. Epub 2016 Dec 1. PubMed PMID: 27916688. 4. Saitoh A, Nagase H. Delta Opioid Receptor (DOR) Ligands and Pharmacology: Development of Indolo- and Quinolinomorphinan Derivatives Based on the Message-Address Concept. Handb Exp Pharmacol. 2016 Oct 28. doi: 10.1007/164_2016_18. [Epub ahead of print] PubMed PMID: 27787711.