TargetMol

Setin-1

Product Code:
 
TAR-T26188
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T26188-100mg100mgEnquire
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
Setin-1 is the most potent Set7 inhibitor that acts by inhibiting the KMTase G9a.
CAS:
1313802-67-3
Formula:
C29H21F3N2O2
Molecular Weight:
486.494
Purity:
0.98
SMILES:
OC(=O)c1cccc(NCc2cccc(c2)-n2ccc3c(cccc23)-c2ccc(cc2)C(F)(F)F)c1

Documents

References

1. Kashyap S, Sandler J, Peters U, Martinez EJ, Kapoor TM. Using 'biased-privileged' scaffolds to identify lysine methyltransferase inhibitors. Bioorg Med Chem. 2014 Apr 1;22(7):2253-60. doi: 10.1016/j.bmc.2014.02.024. Epub 2014 Feb 28. PubMed PMID: 24650704; PubMed Central PMCID: PMC4038709.