TargetMol

CP-122288

Product Code:
 
TAR-T27059
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T27059-5mg5mg£1,091.00
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Quantity:
TAR-T27059-50mg50mg£2,143.00
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Quantity:
TAR-T27059-100mg100mg£2,801.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CP-122288 is a potent and selective agonist for the 5-HT1B, 5-HT1D and 5-HT1F serotonin receptor subtypes. CP-122288 is potent as an inhibitor of plasma protein extravasation and neurogenic inflammation.
CAS:
143321-74-8
Formula:
C16H23N3O2S
Molecular Weight:
321.44
Purity:
0.98
SMILES:
CNS(=O)(=O)Cc1ccc2[nH]cc(C[C@H]3CCCN3C)c2c1

References

1. Roon KI, Olesen J, Diener HC, Ellis P, Hettiarachchi J, Poole PH, Christianssen I, Kleinermans D, Kok JG, Ferrari MD. No acute antimigraine efficacy of CP-122,288, a highly potent inhibitor of neurogenic inflammation: results of two randomized, double-blind, placebo-controlled clinical trials. Ann Neurol. 2000 Feb;47(2):238-41. PubMed PMID: 10665496.