TargetMol

CREBBP-IN-9

Product Code:
 
TAR-T27082
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27082-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T27082-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T27082-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CREBBP-IN-9, a CREBBP inhibitor, acts on the bromodomain of the protein.
CAS:
1219576-50-7
Formula:
C16H15N5O2S
Molecular Weight:
341.39
Purity:
0.98
SMILES:
CC(=O)c1cccc(NC(=O)c2c(C)c(C)sc2-n2cnnn2)c1

References

1. Xu M, Unzue A, Dong J, Spiliotopoulos D, Nevado C, Caflisch A. Discovery of CREBBP Bromodomain Inhibitors by High-Throughput Docking and Hit Optimization Guided by Molecular Dynamics. J Med Chem. 2016 Feb 25;59(4):1340-9. doi: 10.1021/acs.jmedchem.5b00171. Epub 2015 Jul 15. PubMed PMID: 26125948.