TargetMol

Metoprine

Product Code:
 
TAR-T8548
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8548-5mg5mg£115.00
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TAR-T8548-10mg10mg£142.00
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TAR-T8548-1mL1 mL * 10 mM (in DMSO)£149.00
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TAR-T8548-25mg25mg£198.00
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TAR-T8548-50mg50mg£282.00
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TAR-T8548-100mg100mg£389.00
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TAR-T8548-500mg500mg£804.00
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This product comes from: United States.
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Further Information

Bioactivity:
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), with potential antineoplastic activity.
CAS:
7761-45-7
Formula:
C11H10Cl2N4
Molecular Weight:
269.13
Pathway:
Immunology/Inflammation; Cell Cycle/Checkpoint; GPCR/G Protein; Chromatin/Epigenetic; Neuroscience
Purity:
0.9909
SMILES:
Cc1nc(N)nc(N)c1-c1ccc(Cl)c(Cl)c1
Target:
Histone Methyltransferase; Antifolate; Histamine Receptor

Documents

References

Junichi Kitanaka, et al. Brain Histamine N-Methyltransferase As a Possible Target of Treatment for Methamphetamine Overdose. Drug Target Insights. 2016 Mar 2;10:1-7. Samotaeva I S , Birioukova L M , Midzyanovskaya I S , et al. Metoprine induced behavioral modifications and brain regional histamine increase in WAG/Rij and Wistar rats[J]. Epilepsy Research, 2012, 101(1-2):148-156.