TargetMol

BMS-605541

Product Code:
 
TAR-T26852
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26852-5mg5mg£107.00
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Quantity:
TAR-T26852-1mL1 mL * 10 mM (in DMSO)£115.00
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TAR-T26852-10mg10mg£129.00
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TAR-T26852-25mg25mg£197.00
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Quantity:
TAR-T26852-50mg50mg£276.00
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Quantity:
TAR-T26852-100mg100mg£375.00
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Quantity:
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
BMS-605541 is a potent, orally active and selective inhibitor of VEGFR-2.
CAS:
639858-32-5
Formula:
C19H17F2N5OS
Molecular Weight:
401.44
Pathway:
Angiogenesis|Tyrosine Kinase/Adaptors
Purity:
0.98
SMILES:
Fc1cc(F)c(cc1NCc1cnc(Nc2ccccn2)s1)C(=O)NC1CC1
Target:
VEGFR

Documents

References

1. Borzilleri RM, Bhide RS, Barrish JC, D'Arienzo CJ, Derbin GM, Fargnoli J, Hunt JT, Jeyaseelan R Sr, Kamath A, Kukral DW, Marathe P, Mortillo S, Qian L, Tokarski JS, Wautlet BS, Zheng X, Lombardo LJ. Discovery and evaluation of N-cyclopropyl-
2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5- ylmethyl)amino)benzamide (BMS-605541), a selective and orally efficacious inhibitor of vascular endothelial growth factor receptor-2. J Med Chem. 2006 Jun 29;49(13):3766-9. PubMed PMID: 16789733.