TargetMol

YM-58790

Product Code:
 
TAR-T72038
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T72038-1mg1mg£189.00
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TAR-T72038-5mg5mg£330.00
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Quantity:
TAR-T72038-10mg10mg£485.00
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TAR-T72038-25mg25mg£866.00
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Quantity:
TAR-T72038-50mg50mg£1,420.00
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Quantity:
TAR-T72038-100mg100mg£2,238.00
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Quantity:
TAR-T72038-500mg500mg£3,107.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
YM-58790 free base is a potent mAChR antagonist.YM-58790 free base inhibited M1 mAChR, M2 mAChR, and M3 mAChR with Ki values of 28 nM, 260 nM, and 15 nM, respectively.YM-58790 free base inhibits reflex rhythmic bladder contraction in rats by inhibiting bladder pressurization. YM-58790 free base inhibits reflex rhythmic bladder contractions in rats by inhibiting bladder pressurization.
CAS:
168830-70-4
Molecular Weight:
429.55
Pathway:
Neuroscience
Purity:
0.9888
SMILES:
O=C(OC1CCN(CC2=CC=C(C=C2)NC)CC1)NC(C=3C=CC=CC3)C=4C=CC=CC4
Target:
AChR

References

Naito R, et al. Selective muscarinic antagonists. I. Synthesis and antimuscarinic properties of 4-piperidyl benzhydrylcarbamate derivatives. Chem Pharm Bull (Tokyo). 1998 Aug;46(8):1274-85.