TargetMol

PERK-IN-6

Product Code:
 
TAR-T72053
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T72053-1mg1mg£201.00
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TAR-T72053-5mg5mg£388.00
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TAR-T72053-10mg10mg£543.00
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Quantity:
TAR-T72053-25mg25mg£825.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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  • Further Information
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Further Information

Bioactivity:
PERK-IN-6 is a novel and highly potent PERK inhibitor (IC50:2.5 nM).
CAS:
1337532-14-5
Molecular Weight:
398.46
Pathway:
Apoptosis
Purity:
0.9877
SMILES:
O=C(N1C=2C=CC(=CC2CC1)C3=CN(C=4N=CN=C(N)C43)C)CC5=NC(=CC=C5)C
Target:
PERK

Documents

References

Axten JM, et al. Discovery of GSK2656157: An Optimized PERK Inhibitor Selected for Preclinical Development. ACS Med Chem Lett. 2013 Aug 12;4(10):964-8.