TargetMol

EGFR/BRAFV600E-IN-1

Product Code:
 
TAR-T62503
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T62503-100mg100mgEnquire
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TAR-T62503-50mg50mgEnquire
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
EGFR/BRAFV600E-IN-1 (Compound 23) is a potent dual inhibitor of EGFR (IC50: 0.08 uM) and BRAFV600E (IC50: 0.15 uM). EGFR/BRAFV600E-IN-1 exhibited anti-proliferative effects on A-549 (IC50: 1.2 uM), MCF-7 (IC50: 0.79 uM), Panc-1 (IC50: 1.3 uM), HT-29 (IC50: 1.23 uM).
CAS:
2492429-45-3
Molecular Weight:
437.92
Purity:
0.98
SMILES:
Cc1c2C(=O)N(CCc3ccc(cc3)N3CCOCC3)CC(=O)n2c2ccc(Cl)cc12

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