TargetMol

TRK-IN-12

Product Code:
 
TAR-T62531
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T62531-5mg5mg£850.00
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Quantity:
TAR-T62531-50mg50mg£1,661.00
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Quantity:
TAR-T62531-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TRK-IN-12 (Compound 9e) is a potent inhibitor of TRK (TRK G595R IC 50 = 13.1 nM). TRK-IN-12 is a macrocyclic derivative compound. TRK-IN-12 shows significant antiproliferative activity in the Ba/F3-LMNA-NTRK1 cell line ( IC 50 = 0.080 uM). TRK-IN-12 has shown a better inhibitory effect ( IC 50 = 0.646 uM) than control agent LOXO-101 in Ba/F3-LMNA-NTRK1-G595R cell line [1] .
CAS:
2823342-34-1
Molecular Weight:
439.89
Purity:
0.98