TargetMol

(?)-WIN 55,212-3 mesylate

Product Code:
 
TAR-T71963
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T71963-5mg5mg£149.00
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Further Information

Bioactivity:
(-)-WIN 55,212-3 mesylate is an aminoalkylindole derivative which acts as a competitive neutral antagonist of the human cannabinoid CB2 receptor, blocking both the stimulating action of CP 55,940 and the inverse agonism of SR 144528. (-)-WIN 55,212-3 neither antagonizes nor mimics the effects of δ9-THC on rat cerebellar membranes, which presumably express the CB1 receptor. (-)-WIN 55,212-3 also weakly antagonizes the melatonin MT1 and muscarinic M4 receptors but has no effect on several other G protein-coupled receptors.
CAS:
131543-25-4
Molecular Weight:
522.62
Purity:
0.98
SMILES:
CS(O)(=O)=O.Cc1c(C(=O)c2cccc3ccccc23)c2cccc3OC[C@H](CN4CCOCC4)n1c23

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