TargetMol

L 685434

Product Code:
 
TAR-T32463
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T32463-100mg100mgEnquire
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TAR-T32463-500mg500mgEnquire
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
L 685434 is a pseudopeptide that can against HIV protease.
CAS:
126456-36-8
Molecular Weight:
544.692
Purity:
0.98
SMILES:
CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12

Documents

References

Young SD, Payne LS, Thompson WJ, Gaffin N, Lyle TA, Britcher SF, Graham SL, Schultz TH, Deana AA, Darke PL, et al. HIV-1 protease inhibitors based on hydroxyethylene dipeptide isosteres: an investigation into the role of the P1' side chain on structure-activity. J Med Chem. 1992 May 15;35(10):1702-9. PubMed PMID: 1588552. Smith AB 3rd, Hirschmann R, Pasternak A, Yao W, Sprengeler PA, Holloway MK, Kuo LC, Chen Z, Darke PL, Schleif WA. An orally bioavailable pyrrolinone inhibitor of HIV-1 protease: computational analysis and X-ray crystal structure of the enzyme complex. J Med Chem. 1997 Aug 1;40(16):2440-4. PubMed PMID: 9258349.