TargetMol

PROTAC SMARCA2 degrader-7

Product Code:
 
TAR-T89261
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T89261-10mg10mgEnquire
Quantity:
TAR-T89261-50mg50mgEnquire
Quantity:
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This product comes from: Austria.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PROTACSMARCA2 degrader-7 (Compound I-428) is a PROTAC degrader targeting the catalytic subunits SMARCA2 and SMARCA4 of the SWI/SNF complex. In MV411, it achieves degradation of SMARCA2 and SMARCA4 with DC50 values of <100 nM and 100-500 nM, respectively.
CAS Number:
2568277-71-2
Formula:
C50H62N10O5S
Molecular Weight:
915.16
Purity:
98%
SMILES:
C(C12CCC(C(N[C@H](C(=O)N3[C@H](C(NCC4=CC=C(C=C4)C5=C(C)N=CS5)=O)C[C@@H](O)C3)C(C)(C)C)=O)(CC1)CC2)N6CCC(CC6)N7C=C(C=N7)C=8C=C(N=NC8N)C9=C(O)C=CC=C9

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