TargetMol

Erasin

Product Code:
 
TAR-T73472
Product Group:
 
Other Biochemicals
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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This product comes from: Austria.
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Further Information

Bioactivity:
Erasin is a STAT3 inhibitor (IC50 = 9.7 uM) with higher selectivity for inhibiting STAT3 tyrosine phosphorylation than STAT5 and STAT1. It induces apoptosis in various cancer cell lines (e.g., MDA-MB-231, HCC-827) and is effective against Erlotinib-resistant cancer cells.
Formula:
C20H19N3O3
Molwt:
349.38
Pathway:
Stem Cells|JAK/STAT signaling|Apoptosis
SMILES:
CC(C)(C)C1=CC(C2=O)=C(C=C1)OC=C2/C=N/NC(C3=CC=CN=C3)=O
Target:
Apoptosis|STAT

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