TargetMol

CPI1

Product Code:
 
TAR-TP3085
Product Group:
 
Peptides
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-TP3085-10mg10 mgEnquire
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TAR-TP3085-50mg50 mgEnquire
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This product comes from: Austria.
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Further Information

Bioactivity:
CPI1 is an effective and highly specific inhibitor of multidrug resistance protein 1 (MRP1). It exhibits inhibitory activity against MRP1 at the nanomolar level (Ki: 100 nM) and has minimal effect on P-glycoprotein (Pgp). CPI1 competes with LTC4 for binding to the same site on MRP1, inhibiting ATP hydrolysis and substrate transport. It is useful in research related to drug delivery and addressing cancer chemotherapy resistance.
Formula:
C111H131N23O30S
Molwt:
2299.43
Pathway:
Membrane transporter/Ion channel|Neuroscience
SMILES:
C[C@H]([C@H]1C(=O)N[C@@H](CSCC(=O)N[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1)CO)CC(=O)O)CC2=CC=CC=C2)CCC(=O)N)CCC(=O)O)CC3=CC=C(C=C3)O)CC4=CC=C(C=C4)O)CC5=CNC6=CC=CC=C65)CC7=CNC=N7)CC(C)C)CC(=O)N)CC8=CNC9=CC=CC=C98)CC1=CC=CC=C1)CC1=CC=C(C=C1)O)C(=O)O)O
Target:
P-gp

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