TargetMol

GpTx-1 TFA

Product Code:
 
TAR-TP3232
Product Group:
 
Peptides
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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CodeSizePrice
TAR-TP3232-10mg10 mgEnquire
Quantity:
TAR-TP3232-50mg50 mgEnquire
Quantity:
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This product comes from: Austria.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 uM) and NaV1.5 (IC50 = 4.20 uM) with >20-fold and >950-fold selectivity, respectively.
Pathway:
Membrane transporter/Ion channel
Target:
Sodium Channel

Documents