TargetMol

GW590735

Product Code:
 
TAR-T9766
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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This product comes from: Austria.
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Further Information

Bioactivity:
GW590735 is an effective and selective PPARα agonist with an EC50 of 4 nM on PPARα and at least 500-fold selectivity versus PPARδ and PPARγ. GW590735 can be used in dyslipidemia studies.
CAS:
343321-96-0
Formula:
C23H21F3N2O4S
Molecular Weight:
478.48
Pathway:
DNA Damage/DNA Repair; Metabolism
Purity:
0.98
SMILES:
CC(C)(C(O)=O)Oc1ccc(CNC(c2c(C)nc(-c3ccc(C(F)(F)F)cc3)s2)=O)cc1
Target:
PPAR

Documents

References

Sierra ML, et al. Substituted 2-[(4-aminomethyl)phenoxy]-2-methylpropionic acid PPARalpha agonists. Discovery of a novel series of potent HDLc raising agents. J Med Chem. 2007;50(4):685-695.