TargetMol

AChE/BuChE-IN-4

Product Code:
 
TAR-T77758
Product Group:
 
Other Biochemicals
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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This product comes from: Austria.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
AChE/BuChE-IN-4 is a multi-target AChE/BuChE inhibitor with oral activity and blood-brain barrier permeability, with IC50 values of 2.08 and 7.41 uM for AChE and BuChE, respectively.
CAS Number:
1997158-25-4
Formula:
C17H23N5
Molecular Weight:
297.4
Purity:
100%
SMILES:
N=1C=CC(=NC1N)NCC2CCN(CC=3C=CC=CC3)CC2
Target:
AChE

Documents

References

1.Cavdar H,et al. Inhibition of acetylcholinesterase and butyrylcholinesterase with uracil derivatives: kinetic and computational studies. J Enzyme Inhib Med Chem. 2019 Dec;34(1):429-437.